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Urinary antiseptic

Methenamine hippurate

Brand names: Hiprex

Adult dose

Dose: 1g PO BD
Route: PO
Frequency: BD

Clinical pearls

  • Recurrent UTI prophylaxis as alternative to long-term antibiotics (ALTAR trial supports non-inferiority)
  • Requires acidic urine to release formaldehyde

Contraindications

  • Severe hepatic impairment
  • Severe renal impairment
  • Metabolic acidosis
  • Gout (caution — uric acid)

Side effects

  • GI upset
  • Rash
  • Bladder irritation

Interactions

  • Sulphonamides (precipitation)
  • Urinary alkalinisers (reduce activity — needs acidic urine)

Monitoring

  • U&E
  • LFTs

Reference: BNF; NICE NG112; ALTAR trial; https://bnf.nice.org.uk/drugs/methenamine-hippurate/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.