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Ultra-short-acting β1-blocker

Landiolol hydrochloride

Brand names: Rapibloc

Adult dose

Dose: IV: 10–40 micrograms/kg/min infusion; loading possible per BNF/SmPC
Route: IV
Frequency: infusion

Clinical pearls

  • Rapid heart-rate control in supraventricular tachyarrhythmia/peri-operative
  • Half-life ~4 min — easily titratable; cardioselective

Contraindications

  • Severe bradycardia
  • Sick sinus syndrome
  • 2nd/3rd degree AV block
  • Cardiogenic shock
  • Severe hypotension
  • Decompensated heart failure
  • Pulmonary hypertension

Side effects

  • Bradycardia
  • Hypotension
  • Bronchospasm

Interactions

  • Calcium-channel blockers
  • Digoxin
  • Other negative inotropes

Monitoring

  • ECG
  • BP
  • HR continuously

Reference: BNF; ESC; SmPC; https://bnf.nice.org.uk/drugs/landiolol-hydrochloride/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.